Материал: MasterPass _ Pharmacology in 7 Days for Medical Students

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PHARMACOLOGY IN 7 DAYS FOR MEDICAL STUDENTS

•Cyclobarbitone

•Pentobarbitone

iiiShort-acting

•Quinalbarbitone

ivUltrashort-acting

•Methohexitone

•Thiopentone sodium

B Benzodiazepines

iLong-acting

•Chlorazepate

•Diazepam

•Flurazepam

•Nitrazepam

iiIntermediate-acting

•Alprazolam

•Estazolam

•Lorazepam

•Oxazepam

iiiShort-acting

•Lormetazepam

•Triazolam

CNewer agents

iImidazopyridine derivatives

•Zaleplon

•Zolpidem

ii5-HT1A partial agonists

•Buspirone

•Gepirone

•Ipsapirone

DOlder agents

•Chloralhydrate

•Glutethemide

•Meprobamate

•Paraldehyde

Skeletal muscle relaxants

ACentrally-acting muscle relaxants

1Benzodiazepines

•Clorazepate

•Diazepam

•Ketazolam

•Medazepam

2Benzoxazole derivatives

•Benzimidazole

•Chlorzoxazone

•Zoxazolamine

3GABA analogue

•Baclofen

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CLASSIFICATIONS

4Miscellaneous compounds

•Cyclobenzaprine

•Chlormezanone

•Chlorphensin

•Methocarbamol

•Orphenadrine HCl

•Orphendrine citrate

5Propanediol derivatives

•Carisoprodol

•Mephenesin

•Meprobamate

•Styramate

BDirectly-acting muscle relaxants

•Dantrolene

CNeuromuscular blocking agents

iCompetitive blocking/nondepolarising agents

•Alcuronium

•Atracurium

•Dimethyl tubocurarine

•Fazadinium

•Gallamine

•Pancuronium

•Tubocurarine

•Vecuronium

iiDepolarising agents

•Decamethonium

•Suxamethonium

•Suxemethonium

Sulfonamides

1Short-acting (well absorbed by mouth and rapidly eliminated) a General purpose

•Sulfadiazine

•Sulfadimidine

•Sulfamethoxazole

bMainly for UTI

•Sulfamethizole

•Sulfisoxazole

2Long acting (well absorbed by GIT and slowly eliminated)

•Sulfadoxine

•Sulfametopyrazine

•Sulfamethoxypyridazine

•Sulfaphenazole

3Poorly absorbed by GIT

•Sulfaguanidine

•Sulfathalidine

•Succinyl Sulfathiazole

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PHARMACOLOGY IN 7 DAYS FOR MEDICAL STUDENTS

4For topical application

•Sulfacetamide

•Silver Sulfadiazine

5Miscellaneous group

•Sulfapyridine

•Sulfasalazine

6Sulfonamide combinations

•Co-trimoxazole (sulfamethoxazole + trimethoprim)

•Fansidar (sulfadoxine + pyrimethamine)

Tetracyclines

1Based on source a Natural

•Chlortetracycline

•Oxytetracycline

•Demeclocycline b Semi-synthetic

•Clomocycline

•Doxycycline

•Lymecycline

•Minocycline

•Methacycline

•Tetracycline

2Based on duration of action a Short-acting

•Tetracycline

•Chlortetracycline

•Oxytetracycline

•Clomocycline

bIntermediate-acting

•Methacycline

•Lymecycline

•Demeclocycline

cLong-acting

•Doxycycline

•Minocycline

Thiazide diuretics

1Intermediate-acting

•Cyclothiazide

•Methylclothiazide

•Quinethazone

•Trichlormethiazide

2Short-acting

•Bendroflumethiazide

•Cyclopenthiazide

•Chlorothiazide

•Hydrochlorothiazide

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CLASSIFICATIONS

•Hydroflumethiazide

3 Long-acting

•Chlorthalidone

•Indapamide

•Polythiazide

Loop diuretics

1Carboxylic acid derivatives

•Bumetanide

•Furosemide

•Piretanide

•Torsemide

2Phenoxy acetic acid derivatives

•Ethacrynic Acid

•Indacrinone

Antitussives

ADrugs for productive cough

1Expectorants

a Sedative expectorants

iAlkaline expectorants

•Potassium acetate and citrate

iiNauseant expectorants

•Ammonium carbonate and chloride

•Tincture ipecacuanha

iiiSaline expectorants

•Sodium and potassium iodide

bStimulant (aromatic) expectorants

•Creosote

•Guaiacol

•Guaiphenesin

•Terpenehydrate

2Mucolytics

•Ambroxol

•Acetylcysteine

•Bromohexine

•Carbocysteine

•Methylcysteine

•Proteolytic enzymes (e.g. pancreatic domase and trypsin)

B Drugs for unproductive cough

1Peripheral antitussives

a Drugs with local anaesthetic activity

•Benzonatate b Demulcents

•Liquorice lozenges c Steam inhalation

•With tincture menthol

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PHARMACOLOGY IN 7 DAYS FOR MEDICAL STUDENTS

2Central antitussives

a Opioid antitussives

iAddicting drugs

•Dihydromorphinone

•Methadone

•Morphine

iiNon-addicting drugs

•Dihydrocodeinone

•Pholcodine

bNon-opioid antitussives

•Benzonatate

•Carbetapentane

•Chlorphedianol

•Dextromethorphan

•Narcotine

•Oxeladine

Drugs used in cardiac failure

1ACE inhibitors

•Captopril

•Enalapril

•Lisinopril

2Cardiotonic drugs

iβ1-selective adrenoceptor agonists

•Dobutamine

•Prenalterol

iiBipyridine derivatives

•Inamrinone

•Milrinone

iiiCardiac glycosides

•Digoxin

•Digitoxin

•Gitoxin

•Gitaloxin

•Ouabain

•Strophanthin

3Diuretics

iLoop diuretics

•Ethacrynic acid

•Furosemide

iiThiazide diuretics

•Bendrofluazide

•Polythiazide

4Vasodilators

•Hydralazine

•Nifedipine

•Nitroglycerin

•Prazosin

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Источник: https://studfile.net/preview/16445234/