Материал: MasterPass _ Pharmacology in 7 Days for Medical Students

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PHARMACOLOGY IN 7 DAYS FOR MEDICAL STUDENTS

Newer drugs:

1GABA analogue

•Gabapentin

•Vigabatrin

2Miscellaneous

•Lamotrigine

•Felbamate

•Topiramate

Older drugs:

1Bromides

•Sodium and Potassium bromide

2Carbonic anhydrase inhibitors

•Acetazolamide

3Oxazolidinedione derivatives

•Trimethadione

4Miscellaneous

•Paraldehyde

Adrenocorticosteroids

Natural

1Glucocorticoids

•Cortisol

•Corticosterone

2Mineralocorticoids

•Aldosterone

•11-Deoxy corticosterone acetate

Synthetic

1Glucocorticoids

•Cortisone

•Prednisone

•Prednisolone

•Methylprednisolone

•Paramethasone

•Dexamethasone

•Triamcinolone

•Betamethasone valerate

•Beclomethasone dipropionate

2Mineralocorticoids

1 Fludrocortisone

Antiviral drugs

1Agents to treat herpes simplex virus (HSV) and varicella-zoster virus (VSV) infections (DNA-polymerase inhibitors)

•Acyclovir

•Valacyclovir

•Famciclovir

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CLASSIFICATIONS

•Penciclovir

•Foscarnet

•Trifluridine

2Agents to treat cytomegalovirus (CMV) infections

•Cidofovir

•Foscarnet

•Fomivirsen

•Ganciclovir

•Valganciclovir

3Antiretroviral agents

iNucleoside reverse transcriptase inhibitors (NRTIs)

•Abacavir

•Didanosine

•Lamivudine

•Stavudine

•Zidovudine

•Zalcitabine

iiNon-nucleoside reverse transcriptase inhibitors (NNRTIs)

•Delavirdine

•Efavirenz

•Nevirapine

iiiProtease inhibitors

•Amprenavir

•Indinavir

•Nelfinavir

•Ritonavir

•Saquinavir

ivFusion inhibitors

•Enfuvirtide

4Antihepatitis agents

•Adefovir

•Interferon

•Lamivudine

•Ribavirin

5Anti-influenza agents

•Amantadine

•Rimantadine

•Oseltamivir

•Zanamivir

NSAIDs

ADrugs with analgesic and marked anti-inflammatory effects

1Salicylic acid derivatives

•Aspirin (acetyl salicylic acid)

•Salicylic acid

•Sodium salicylate

•Methyl salicylate

•Choline salicylate

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PHARMACOLOGY IN 7 DAYS FOR MEDICAL STUDENTS

•Magnesium salicylate

•Diflunisal

•Benorylate

2Pyrazolone derivatives

•Phenylbutazone

•Oxyphenbutazone

•Azapropazone

3Acetic acid derivatives

•Diclofenac

•Indomethacin

•Tolmetin

•Sulnidac

•Etodolac

4Oxicams

•Piroxicam

•Meloxicam

5Miscellaneous

•Nimuselide

•Celecoxib

•Rofecoxib

BDrugs with analgesic and moderate anti-inflammatory effects

1Propionic acid derivatives

•Ibuprofen

•Ketoprofen

•Fenoprofen

•Flurbiprofen

•Carprofen

•Indoprofen

•Naproxen

•Oxaprozin

2Fenamic acid derivatives

•Mefenamic acid

•Meclofenamic acid

•Flufenamic acid

•Tolfenamic acid

CDrugs with analgesic and weak anti-inflammatory effects

•Paracetamol (aniline derivative)

Adrenergic neuron blockers

1Drugs which interfere with synthesis of noradrenaline

•Metyrosine (alpha-methyl tyrosine)

2Drugs that inhibit storage of noradrenaline

•Deserpidine

•Reserpine

3Drugs that prevent release of noradrenaline

•Bethanidine

•Debrisoquin

•Guanadrel

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CLASSIFICATIONS

•Guanethidine

•Guanoxan

Alpha-adrenergic blockers

AChemical classification

1Beta-haloalkylamines

•Dibenamine

•Phenoxybenzamine

2Benzodioxans

•Dibuzaine

•Diperoxan

3Benzene sulfonamide

•Tamsulosin

4Dibenzapines

•Azepetine

5Ergot alkaloid

•Dihydroergotamine

•Ergotamine

6Phenothiazines

•Chlorpromazine

7Phenoxyalkylamines

•Thymoxamine

8Piperazinyl quinazolines

•Doxazosin

•Prazosin

•Terazosin

9Substituted imidazolines

•Phentolamine

•Tolazoline

10Miscellaneous

•Carvedilol

•Indoramin

•Labetalol

BAccording to reversibility of action

1Irreversible (non-competitive blockers; long-acting)

•Dibenamine

•Phenoxybenzamine

2Reversible (competitive blockers; short-acting)

•Doxazosin

•Prazosin

•Phentolamine

•Terazosin

•Tolazoline

•Trimazosin

•Urapidil

CAccording to receptor selectivity

1Mixed α and β adrenoceptor blocking drugs

•Carvedilol

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PHARMACOLOGY IN 7 DAYS FOR MEDICAL STUDENTS

• Labetalol

2Selective α-blockers

iα1-blockers

•Alfuzosin

•Doxazosin

•Pinacidal

•Prazosin

•Tamsulosin

•Teruzosin

•Trimazosin

iiα2-blockers

•Idazoxan

•Yohimbine

3Non-selective (both α1 and α2-blockers)

•Dibenamine

•Dihydroergotamine

•Ergotamine

•Phentolamine

•Phenoxybenzamine

•Tolazoline

Aminoglycosides

1Natural

•Gentamycin

•Kanamycin

•Neomycin

•Streptomycin

•Tobramycin

2Semi-synthetic

•Amikacin

•Netilmicin

Members of macrolide group

•Azithromycin

•Clarithromycin

•Roxithromycin

•Telithromycin

•Carbomycin

•Erythromycin

•Oleandomycin

•Spiramycin

Amoebicides

AChemical classification

1Dichloroacetamides

•Clefamide

•Etofamide

•Diloxanide furoate

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Источник: https://studfile.net/preview/16445234/