Материал: MasterPass _ Pharmacology in 7 Days for Medical Students

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PHARMACOLOGY IN 7 DAYS FOR MEDICAL STUDENTS

eOthers

•Bupropion

•Trazodone

5 Miscellaneous

• Alprazolam

• Flupenthixol

Antidiarrhoeal drugs

1Antimotility agents (drugs that prolong intestinal transit time by reducing motility)

a Anticholinergics

•Atropine

•Dicyclomine HCl

•Propantheline

bBismuth subsalicylate

cNaturally occurring opium alkaloids

•Codeine phosphate

dSynthetic opioid compounds

•Diphenoxylate

•Loperamide

2Adsorbants

•Chalk

•Charcoal

•Isphagol husk

•Kaolin

•Methyl cellulose

•Pectin

3Miscellaneous

•Peppermint oil

•Vegetable astringent

Anti-emetics

1Anticholinergics

•Hyoscine

2Antihistamines (H1-antagonists)

•Cyclizine

•Hydroxyzine

•Meclizine

•Promethazine

•Dimenhydrinate

•Diphenhydramine

3Benzodiazepines

•Diazepam

4Cannabinoids

•Dronabinol

•Nabilone

5D2-receptor antagonists

•Domperidone

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CLASSIFICATIONS

•Metoclopramide

6 Glucocorticoids

•Dexamethasone

•Methylprednisolone

7Neurokinin-I-receptor-antagonists

•Aprepitant

8Phenothiazines

•Chlorpromazine

•Prochlorperazine

•Thiethylperazine

9Selective 5-HT3 receptor antagonists

•Dolasetron

•Granisetron

•Ondansetron

•Palonosetron

Antifungal drugs

1Drugs that disrupt fungal cell membrane A Polyenes

•Amphotericin

•Nystatin

BAzoles

iImidazoles

•Ketoconazole

iiTriazoles

•Fluconazole

iiiAllylamines

•Terbinafine

2Drug that inhibits mitosis

•Griseofulvin

3Drug that inhibits DNA synthesis

•Flucytosine

Antimalarial drugs

AChemical classification

1Cinchona alkaloids

•Quinine

2Diaminopyrimidine

•Pyrimethamine

3Folate antagonists

•Proguanil

44-Aminoquinolines

•Amodiaquine

•Chloroquine

58-Aminoquinolines

•Primaquine

6Quinoline methanol

•Mefloquine

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PHARMACOLOGY IN 7 DAYS FOR MEDICAL STUDENTS

• Quinidine

7Sulfonamides

•Sulphadoxine

8Sulphones

•Dapsone

9Tetracyclines

•Doxycycline

10Miscellaneous

•Halofantrin

•Qinghaosu derivatives (artemisinins), i.e. artemether and artisunate

11Combinations

•Fansidar (pyrimethamine + sulfadoxine)

•Fansimef (pyrimethamine + sulfadoxine + mefloquine)

•Maloprim (pyrimethamine + dapsone)

•Malarone (atovaquone + proguanil)

BClassification based on site of action

1Tissue schizonticides (acting on hepatic cycle: pre-erythrocytic stage) a Against primary tissue forms for causal prophylaxis

• Proguanil

bAgainst latent tissue forms, for terminal prophylaxis/radical cure

•Primaquine

2Blood schizonticides (acting on erythrocytic cycle for suppressive cure) a Rapidly acting blood schizonticides

•Artemisinins

•Amodiaquine

•Chloroquine

•Halofantrin

•Mefloquine

•Quinine

bSlower acting blood schizonticides

•Doxycycline

•Proguanil

•Pyrimethamine

3Gametocides against sexual erythrocytic forms

•Primaquine (against plasmodium falciparum)

•Chloroquine and quinine (against plasmodium vivax and ovale)

Antigout drugs

ADrugs for acute attack

1Natural alkaloids

•Colchicine

•Demecolchicine

2NSAIDs specially used in gout

•Fenoprofen

•Indomethacine

•Naproxen

•Oxaprozin

•Oxyphenbutazone

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CLASSIFICATIONS

•Phenylbutazone

•Piroxicam

3Corticosteroids

•Hydrocortisone

•Prednisolone

BDrugs for chronic gout

1Drugs which increase excretion of uric acid (uricosuric agents)

•Aspirin (in high doses)

•Oxyphenbutazone

•Phenylbutazone

•Probenecid

•Sulfinpyrazone

2Drugs which decrease synthesis of uric acid (xanthine oxidase inhibitors)

•Allopurinol

Antihelminthic drugs

1Drugs acting against nematodes

•Albendazole

•Mebendazole

•Thiabendazole

•Diethyl carbamazine

•Pyrantel pamoate

2Drugs acting against trematodes

•Praziquantel

3Drugs acting against cestodes

•Niclosamide

Drugs used in the Rx of leprosy

•Clofazimine

•Dapsone

•Fluoroquinolones

•Macrolides

•Minocycline

•Rifampicin

•Miscellaneous:

–Ethionamide

–Thalidomide

Drugs used in the Rx of tuberculosis

1First-line drugs

•Ethambutol

•Isoniazid

•Pyrazinamide

•Rifampin

•Streptomycin

2Second-line drugs

•Alikacin and kanamycin

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PHARMACOLOGY IN 7 DAYS FOR MEDICAL STUDENTS

•Ciprofloxacin, levofloxacin and ofloxacin

•Capreomycin

•Cycloserine

•Ethionamide

•Rifabutin

•Rifapentine

Antihypertensive drugs

ACalcium channel blockers

1Benzothiazepines

•Diltiazem

2Diarylaminopropylamine

•Bepridil

3Dihydropyridines

•Amlodipine

•Felodipine

•Isradipine

•Nicardipine

•Nifedipine

•Nimodipine

•Nisoldipine

•Nitrendipine

4Diphenylpiperazines

•Flunarizine

•Ranolazine

•Trimetazidine

5Phenyl Alkylamines

•Gallopamil

•Verapamil

BDiuretics

1Loop diuretics

•Bumetanide

•Ethacrynic acid

•Furosemide

2Potassium-sparing diuretics

•Amiloride

•Spironolactone

•Triamterene

3Thiazides and related agents

•Benzthiazide

•Chlorthalidone

•Chlorothiazide

•Hydrochlorothiazide

•Indapamide

CDrugs acting on renin-angiotensin system

1Angiotensin converting enzyme (ACE) inhibitors

•Benzapril

•Captopril

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Источник: https://studfile.net/preview/16445234/